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Bioorganic synthesis of a recombinant HIV-1 fusion inhibitor, SC35EK, with an N-terminal pyroglutamate capping group Kajiwara, Kazumi, Watanabe, Kentaro, Tokiwa, Rei, Kurose, Tomoko, Ohno, Hiroaki, Tsutsumi, Hiroko, Hata, Yoji, Izumi, Kazuki, Kodama, Eiichi, Matsuoka, Masao, Oishi, Shinya, Fujii, Nobutaka (2009-12-01) Bioorganic & medicinal chemistry, 17(23): 7964-7970 | ![]() |
Affinity selection and sequence-activity relationships of HIV-1 membrane fusion inhibitors directed at the drug-resistant variants Oishi, Shinya, Watanabe, Kentaro, Ito, Saori, Tanaka, Michinori, Nishikawa, Hiroki, Ohno, Hiroaki, Shimane, Kazuki, Izumi, Kazuki, Sakagami, Yasuko, Kodama, Eiichi N., Matsuoka, Masao, Asai, Akira, Fujii, Nobutaka (2010) MedChemComm, 1(4): 276-281 | ![]() |
Design and synthesis of a novel class of CK2 inhibitors: application of copper- and gold-catalysed cascade reactions for fused nitrogen heterocycles Suzuki, Yamato, Oishi, Shinya, Takei, Yoshinori, Yasue, Misato, Misu, Ryosuke, Naoe, Saori, Hou, Zengye, Kure, Tatsuhide, Nakanishi, Isao, Ohno, Hiroaki, Hirasawa, Akira, Tsujimoto, Gozoh, Fujii, Nobutaka (2012-04-25) Organic & biomolecular chemistry, 10(25): 4907-4915 | ![]() |
Development and application of fluorescent SDF-1 derivatives Masuda, Ryo, Oishi, Shinya, Tanahara, Noriko, Ohno, Hiroaki, Hirasawa, Akira, Tsujimoto, Gozoh, Kodama, Eiichi, Matsuoka, Masao, Fujii, Nobutaka (2012-05) Future medicinal chemistry, 4(7): 837-844 | ![]() |
Structure-activity relationship study of tachykinin peptides for the development of novel neurokinin-3 receptor selective agonists Misu, Ryosuke, Noguchi, Taro, Ohno, Hiroaki, Oishi, Shinya, Fujii, Nobutaka (2013-04-15) Bioorganic & medicinal chemistry, 21(8): 2413-2417 | ![]() |
Synthesis and functional analysis of deferriferrichrysin derivatives: Application to colorimetric pH indicators Kobayashi, Yuka, Oishi, Shinya, Kobayashi, Kazuya, Ohno, Hiroaki, Tsutsumi, Hiroko, Hata, Yoji, Fujii, Nobutaka (2013-07-15) Bioorganic & medicinal chemistry, 21(14): 4296-4300 | ![]() |
Affinity-based screening of MDM2/MDMX-p53 interaction inhibitors by chemical array: Identification of novel peptidic inhibitors Noguchi, Taro, Oishi, Shinya, Honda, Kaori, Kondoh, Yasumitsu, Saito, Tamio, Kubo, Tatsuhiko, Kaneda, Masato, Ohno, Hiroaki, Osada, Hiroyuki, Fujii, Nobutaka (2013-07-01) Bioorganic & medicinal chemistry letters, 23(13): 3802-3805 | ![]() |
Concise synthesis and anti-HIV activity of pyrimido[1,2-c][1,3]benzothiazin-6-imines and related tricyclic heterocycles Mizuhara, Tsukasa, Oishi, Shinya, Ohno, Hiroaki, Shimura, Kazuya, Matsuoka, Masao, Fujii, Nobutaka (2012-06-22) Organic & biomolecular chemistry, 10(33): 6792-6802 | ![]() |
Structure-activity relationship study of pyrimido[1,2-c][1,3]benzothiazin-6-imine derivatives for potent anti-HIV agents Mizuhara, Tsukasa, Oishi, Shinya, Ohno, Hiroaki, Shimura, Kazuya, Matsuoka, Masao, Fujii, Nobutaka (2012-11-01) Bioorganic & medicinal chemistry, 20(21): 6434-6441 | ![]() |
Lewis-acid-mediated ring-exchange reaction of dihydrobenzofurans and its application to the formal total synthesis of (−)-quinocarcinamide Chiba, Hiroaki, Sakai, Yuki, Oishi, Shinya, Fujii, Nobutaka, Ohno, Hiroaki (2012-11) Tetrahedron Letters, 53(46): 6273-6276 | ![]() |
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