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Identification of anti-HIV agents with a novel benzo[4,5]isothiazolo[2,3-a]pyrimidine scaffold Okazaki, Shiho, Mizuhara, Tsukasa, Shimura, Kazuya, Murayama, Hiroto, Ohno, Hiroaki, Oishi, Shinya, Matsuoka, Masao, Fujii, Nobutaka (2015-04-01) Bioorganic & medicinal chemistry, 23(7): 1447-1452 | ![]() |
Design and synthesis of biotin- or alkyne-conjugated photoaffinity probes for studying the target molecules of PD 404182 Mizuhara, Tsukasa, Oishi, Shinya, Ohno, Hiroaki, Shimura, Kazuya, Matsuoka, Masao, Fujii, Nobutaka (2013-04) Bioorganic & medicinal chemistry, 21(7): 2079-2087 | ![]() |
Identification of minimal sequence for HIV-1 fusion inhibitors Nishikawa, Hiroki, Oishi, Shinya, Fujita, Mizuno, Watanabe, Kentaro, Tokiwa, Rei, Ohno, Hiroaki, Kodama, Eiichi, Izumi, Kazuki, Kajiwara, Keiko, Naitoh, Takeshi, Matsuoka, Masao, Otaka, Akira, Fujii, Nobutaka (2008-10-15) Bioorganic & medicinal chemistry, 16(20): 9184-9187 | ![]() |
Bioorganic synthesis of a recombinant HIV-1 fusion inhibitor, SC35EK, with an N-terminal pyroglutamate capping group Kajiwara, Kazumi, Watanabe, Kentaro, Tokiwa, Rei, Kurose, Tomoko, Ohno, Hiroaki, Tsutsumi, Hiroko, Hata, Yoji, Izumi, Kazuki, Kodama, Eiichi, Matsuoka, Masao, Oishi, Shinya, Fujii, Nobutaka (2009-12-01) Bioorganic & medicinal chemistry, 17(23): 7964-7970 | ![]() |
Affinity selection and sequence-activity relationships of HIV-1 membrane fusion inhibitors directed at the drug-resistant variants Oishi, Shinya, Watanabe, Kentaro, Ito, Saori, Tanaka, Michinori, Nishikawa, Hiroki, Ohno, Hiroaki, Shimane, Kazuki, Izumi, Kazuki, Sakagami, Yasuko, Kodama, Eiichi N., Matsuoka, Masao, Asai, Akira, Fujii, Nobutaka (2010) MedChemComm, 1(4): 276-281 | ![]() |
Development and application of fluorescent SDF-1 derivatives Masuda, Ryo, Oishi, Shinya, Tanahara, Noriko, Ohno, Hiroaki, Hirasawa, Akira, Tsujimoto, Gozoh, Kodama, Eiichi, Matsuoka, Masao, Fujii, Nobutaka (2012-05) Future medicinal chemistry, 4(7): 837-844 | ![]() |
Concise synthesis and anti-HIV activity of pyrimido[1,2-c][1,3]benzothiazin-6-imines and related tricyclic heterocycles Mizuhara, Tsukasa, Oishi, Shinya, Ohno, Hiroaki, Shimura, Kazuya, Matsuoka, Masao, Fujii, Nobutaka (2012-06-22) Organic & biomolecular chemistry, 10(33): 6792-6802 | ![]() |
Structure-activity relationship study of pyrimido[1,2-c][1,3]benzothiazin-6-imine derivatives for potent anti-HIV agents Mizuhara, Tsukasa, Oishi, Shinya, Ohno, Hiroaki, Shimura, Kazuya, Matsuoka, Masao, Fujii, Nobutaka (2012-11-01) Bioorganic & medicinal chemistry, 20(21): 6434-6441 | ![]() |
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